计算溶液所需的质量、体积或浓度。
| 活性类型 | 活性值-log(M) | 作用机制 | 期刊 | 参考文献(PubMed IDs) |
|---|
| 货号 (SKU) | 包装规格 | 是否现货 | 价格 | 数量 |
|---|---|---|---|---|
| S655396-1ml |
1ml |
期货 ![]() |
|
| 规格或纯度 | 10mM in DMSO |
|---|---|
| 英文名称 | SAFit1 |
| 生化机理 | SAFit1 是一种 FK506 结合蛋白 51 ( FKBP51 )特异性抑制剂,其 K i 为 4±0.3 nM。 |
| 储存温度 | -80℃储存 |
| 运输条件 | 超低温冰袋运输 |
| 产品介绍 |
SAFit1 is a FK506 binding protein 51 ( FKBP51 )-specific inhibitor with a K i of 4±0.3 nM In Vitro SAFit1 (1-1000 nM) potently stimulates neurite outgrowth in two neuronal cell lines (N2a and SH-SY5Y) as well as in primary hippocampal neurons. SAFit1 is active over a wide concentration range. MCE has not independently confirmed the accuracy of these methods. They are for reference only. IC50& Target:Ki: 4±0.3 nM (FKBP51), >50000 nM (FKBP52) |
| Canonical SMILES | COC1=C(C=C(C=C1)CCC(C2=CC(=CC=C2)OCC(=O)O)OC(=O)C3CCCCN3C(=O)C(C4CCCCC4)C5=CC(=C(C(=C5)OC)OC)OC)OC |
|---|---|
| 分子量 | 747.87 |